From: In vitro microbiological evaluation of 1,1'-(5,5'-(1,4-phenylene)bis(3-aryl-1H-pyrazole-5,1-(4H,5H)-diyl))diethanones, novel bis acetylated pyrazoles
Compounds
M. Tuberculosis H37Rv
INH resistant M. tuberculosis
1.00 (μg/mL)
2.00 (μg/mL)
7
74
78
73
77
8
85
89
79
82
9
10
81
80
11
83
12
84
Isoniazid
99
90
96