Compound code
|
R
|
R
1
|
Yield (%)
|
Compound code
|
R
|
R
1
|
Yield (%)
|
---|
3a
|
H
|
|
82
|
3 g
|
4-Cl
|
|
81
|
3b
|
H
|
|
80
|
3 h
|
4-Cl
|
|
83
|
3c
|
H
|
|
82
|
3i
|
4-Cl
|
|
83
|
3d
|
4-F
|
|
84
|
3j
|
2-Cl
|
|
83
|
3e
|
4-F
|
|
86
|
3 k
|
2-Cl
|
|
80
|
3f
|
4-F
|
|
84
|
3 l
|
2-Cl
|
|
86
|
- R, substitution on the phenyl ring; R1, substituted cyclic amine (as depicted in Scheme 1).